1-Boc-3-(Amino)azetidine CAS NO.193269-78-2

Lorcaserin(856681-05-5)is an orally administered agent and a selective 5-HT2C receptor agonist for the treatment of obesity. It had been approved for marketing in US by FDA on 27 June in 2012. In clinical studies, lorcaserin has demonstrated efficacy in obese and overweight populations by promoting weight loss and improving metabolic parameters, and it is well tolerated.

Details

Product Name:	1-Boc-3-(Amino)azetidine
Synonyms:	3-AMINO-1-N-BOC-AZETIDINE;3-AMINO-1-BOC-AZETIDINE;3-AMINO-AZETIDINE-1-CARBOXYLIC ACID TERT-BUTYL ESTER;3-AMINO-AZETIDINE-1-CARBOXYLIC ACID TERT-BUTYL ESTER HYDROCHLORIDE;3-AMINOAZETIDINE, N1-BOC PROTECTED;1-BOC-3-(AMINO)AZETIDINE;1-BOC-3-AMINOAZETIDINE HYDROCHLORIDE;TERT-BUTYL 3-AMINOAZETIDINE-1-CARBOXYLATE
CAS:	193269-78-2
MF:	C8H16N2O2
MW:	172.22
EINECS:
Product Categories:	pharmacetical;Heterocycles series;Amines;Azetidine;Heterocyclic Compounds;Ring Systems;Heterocycles;Miscellaneous Reagents
Mol File:	193269-78-2.mol

1-Boc-3-(Amino)azetidine Chemical Properties

bp	79-81 3mm
storage temp.	Refrigerator
CAS DataBase Reference	193269-78-2(CAS DataBase Reference)

Safety Information

Hazard Codes	Xi,Xn
Risk Statements	34-51-22
Safety Statements	26-36
RIDADR	2735
Hazard Note	Irritant
HazardClass	IRRITANT

MSDS Information

 

1-Boc-3-(Amino)azetidine Usage And Synthesis

Chemical Properties

Clear Colourless to Pale Yellow Oil

1-Boc-3-(Amino)azetidine Preparation Products And Raw materials

Raw materials

Etanol-->Ethyl acetate-->Methanol-->N,N-Dimethylformamide-->Toluene-->Triethylamine-->Palladium-->1,4-Dioxane-->Dimethyl sulfoxide-->Di-tert-butyl dicarbonate-->Xylene-->Hydrazine hydrate-->Triphenylphosphine-->Potassium iodide-->Iodine-->Epichlorohydrin-->Methanesulfonyl chloride-->Imidazole-->Citric acid-->Potassium phthalimide-->3-Hydroxyazetidine hydrochloride-->Aminodiphenylmethane-->Cetyltributylphosphonium bromide